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POST-DOCTORAL RESEARCH FELLOW

Elucidation of substrate recognition and reaction mechanism in the
methyltransferases of cobalamin biosynthesis

A BBSRC-funded postdoctoral post is available immediately, for 3 years, to
elucidate the structures of methyltransferases both free and in complex with
their tetrapyrrole substrates.  The methyltransferases catalyse no fewer than
six of the 30 enzyme-mediated steps in the biosynthesis of vitamin B12
(cobalamin) from 5-aminolevulinic acid. These methylations prevent reversible
C-protonation and leads to the formation of particular tautomeric
intermediates. The specific spatial and temporal addition of the eight
methylations on the macrocycle reveals the importance of forming the correct
double bond configurations essential for much of the chemistry that is required
for corrin ring synthesis. The coupling of methylation and ring contraction is
an exemplar. The post is mainly concerned with the crystallization and X-ray
crystal structure determination of the enzymes and complexes and some of the
enzymes have already been crystallized.  There are also opportunities to be
involved in the production of enzymes and tetrapyrrole intermediates, and
thermodynamic and kinetic analyses. Crystallization of the oxygen-sensitive
intermediates will make use of anaerobic crystallization facilities. A PhD in a
relevant subject area and a strong research background in protein
crystallography and protein chemistry are required. Application deadline 3
November 2006. The post is based at Queen Mary, University of London.

Informal enquiries to: Prof Richard Pickersgill, tel: +44 (0)20 78826360,
email: [EMAIL PROTECTED] or Prof. Martin Warren, tel: +44 (0)1227
824690, email:[EMAIL PROTECTED]

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Richard W Pickersgill
School of Biological and Chemical Sciences
Queen Mary, University of London
Mile End Road
London E1 4NS

T: 02078826360
F: 02089830973
E: [EMAIL PROTECTED]
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