>   Here you are starting to mix equilibrium arguments with the previous
kinetic arguments. 

I don't think I am mixing them; both are relevant. If it cannot diffuse
there, forget the kinetics - necessary but not sufficient requirement.
Nonetheless, the fact that in high concentrations you can force even weak
non-native binders into binding sites (but I reiterate, never in 100%
occupancy, at best asymptotically approaching it) is the reason for the many
buffer 'ligands' observed in structures (also basis for fragment screening.)

>   Your movie doesn't include any details of concentration of your dye, nor
what its binding constant is to any sites in a protein nor any mention of
kon or koff.

The movie does not claim to be a study of any specific ligand binding, it
simply illustrates soaking. Graphs of concentration vs achievable
equilibrium occupancy at different Kds are in separate figures eg 3-40. 

Cheers, BR

Dale Tronrud


> 
> -----Original Message-----
> From: CCP4 bulletin board [mailto:[email protected]] On Behalf Of 
> Keller, Jacob
> Sent: Friday, June 27, 2014 3:07 PM
> To: [email protected]
> Subject: Re: [ccp4bb] Solvent channels
> 
> ....And yet halides--even iodide--permeate those same lysozyme 
> crystals and others entirely in <30--60 sec.
> 
> JPK
> 
> -----Original Message-----
> From: CCP4 bulletin board [mailto:[email protected]] On Behalf Of 
> Bernhard Rupp
> Sent: Friday, June 27, 2014 9:00 AM
> To: [email protected]
> Subject: Re: [ccp4bb] Solvent channels
> 
> Just a remark: diffusion is a slow and random-walk process. 
> Particularly large molecules in viscous media (PEG anybody?) move 
> (diffuse) slowly in solution. To simply extrapolate from the fact that 
> the ligand is smaller than the solvent channels to the odds of the 
> presence of a ligand is a risky proposition. Positive omit difference 
> density after 'shoot first' as Boaz indicated is a much better indication.
And shoot you probably will a lot.
> 
> The little movie below shows how slowly even a small aromatic dye 
> molecule soaks into a crystal.  Total time 10 hrs.
> 
> http://www.ruppweb.org/cryscam/lysozyme_dye_small.wmv
> 
> The literally hundreds of empty ligand structures collected in 
> Twilight attest to that fact.
> 
> http://journals.iucr.org/d/issues/2013/02/00/issconts.html
> 
> Best, BR
> 
> Science is a way of trying not to fool yourself: The first principle 
> is that you must not fool yourself - and you are the easiest person to
fool.
> 
> R. Feynman, 1974
> 
> -----Original Message-----
> From: CCP4 bulletin board [mailto:[email protected]] On Behalf Of 
> Boaz Shaanan
> Sent: Friday, June 27, 2014 2:26 PM
> To: [email protected]
> Subject: Re: [ccp4bb] Solvent channels
> 
> Hi,
> 
> I'm not aware of a program with an option to display channels in 
> crystals but if you use any of the currently available molecular 
> display program and ask to display symmetry-related molecules + 
> adjacent unit cells, it should give you a good enough idea of the 
> spaces between molecules. Using programs for calculation of intermolecular
distances would also be helpful here.
> Independently of the calculation, I would try soaking first and 
> consult the calculations later (in the spirit of Rossmann's American 
> method: shoot first ask later).
> 
>   Cheers,
> 
>            Boaz
> 
> 
> Boaz Shaanan, Ph.D.
> Dept. of Life Sciences
> Ben-Gurion University of the Negev
> Beer-Sheva 84105
> Israel
> 
> E-mail: [email protected]
> Phone: 972-8-647-2220  Skype: boaz.shaanan
> Fax:   972-8-647-2992 or 972-8-646-1710
> 
> 
> 
> 
> 
> ________________________________________
> From: CCP4 bulletin board [[email protected]] on behalf of Reza 
> Khayat [[email protected]]
> Sent: Friday, June 27, 2014 2:00 PM
> To: [email protected]
> Subject: [ccp4bb] Solvent channels
> 
> Hi,
> 
> I'd like to do some soaking experiments with a relatively large molecule.
> Can someone suggest a program/method to display the solvent channels 
> of a crystal? We have the crystal structure. I'd like to see if the 
> channels are large enough to allow the molecule to travel to the 
> hypothesized binding site.
> Thanks.
> 
> Best wishes,
> Reza
> 
> Reza Khayat, PhD
> Assistant Professor
> The City College of New York
> Department of Chemistry, MR-1135
> 160 Convent Avenue
> New York, NY  10031
> Tel. (212) 650-6070
> www.khayatlab.org
> =
> 

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