Dear Monica,

here are some comments from my side:
-one can ask the bulletin board, or just decrease the occupancy during 
refinement and see what happens. If the statistics get better: keep it, if they 
get worse: reject the result.
-I think it is not a question of correct or incorrect structures. You have two 
structures: one with a short soak and low ligand concentration, and one with a 
longer soak and higher ligand concentration, but with 88% complete data. I 
would refine both structures independently and in both cases refine a group 
occupancy for the ligand. If this is done correctly, I would expect that both 
structures will look very similar and provide independent proof for the binding 
mode of your ligand. One question is: what to do with ambiguities in the 
low-occupancy structure? I would look in the high-occupancy structure for hints 
how to resolve these, but more puritan crystallographers may have different 
opinions. Also 88% completeness is not great, but also not that bad. If the 
electron density looks good, I would trust it.

However, if both independently refined structures show a very different binding 
mode, I would get suspicious. In this case I would not just ignore the 
low-occupancy structure but would try to find out what happened: was the ligand 
incorrectly fitted? Where the soaking conditions (precipitant, buffer, pH) 
different, could it be that the ligand was degraded/turned over during the long 
soak?

Best,
Herman

Von: CCP4 bulletin board [mailto:[email protected]] Im Auftrag von Monica 
Mittal
Gesendet: Mittwoch, 13. August 2014 07:48
An: [email protected]
Betreff: [ccp4bb] Protein_Ligand Suggestion

Dear all

I have solved a structure of protein with ligand at 2.7 and 2.8 A. Both have 
ligand bound in it as i soaked it.

For the first structure i soaked for lesser time and lesser concentration of 
ligand and solved it at 2.7 A resolution. Although the ligand has good density 
(2Fo-Fc at 0.9 sigma) but it is little unconnected from its middle portion. Its 
RSCC value is 0.76 and B-factor of 70.0. Overall completeness of structure is > 
91%. So If i decrease the occupancy of ligand here, will it improve the ligand 
statistics esp. the Real space R-value??

However for the second structure, i soaked for longer time and higher ligand 
concentration, so the ligand is perfect with clear 2Fo-Fc map at 1.2 sigma and 
Fo-Fc map at 2.8 sigma along with well defined simulated annealing and 
composite omit maps. The RSCC value is 0.81 with B-factor of 40.1.The only 
issue is the overall completeness of the structure is 88%. But if i get 
evrything OK at this completeness, den can i consider the second structure with 
ligand as the correct one??

Thanks in advance.
Monica

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