Dear Jessica,

The Small Molecule Drug Discovery Suite and the Software "Maestro" of 
Schrödinger could be very useful. But it is not free.

https://www.schrodinger.com/suites/small-molecule-drug-discovery-suite


You could map or predict binding sites of your protein of interest and 
determine which amino acids could be part of the binding pocket. However, I 
don't think it will be considered a quantitative description of the binding 
pocket, because you will be using a static conformation of the protein if you 
use a crystal structure from the PDB. You could also try molecular docking and 
MM-GBSA calculations to predict which residues could interact with the ligand 
and indirectly quantify the electrostatic and hydrophobic contribution from 
each amino acid.


Best,

Pedro De la Torre.
Sotomayor Lab.
________________________________
From: CCP4 bulletin board <[email protected]> on behalf of Jessica M. 
Carpenter <[email protected]>
Sent: Tuesday, June 11, 2019 4:02 PM
To: [email protected]
Subject: [ccp4bb] Characterizing a binding pocket


Dear all,



Can any of you recommend softwares/web servers/programs to calculate the 
volume, hydrophobicity, and electrostatics of a binding pocket in a protein 
structure?  I am trying to quantitatively describe the heme binding pocket of a 
protein by characterizing the residues surfacing the pocket/cavity. Thank you 
very much.



Jessica Carpenter



Graduate student

Department of Chemistry

Dartmouth College

Hanover, NH 03755

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