Thanks for the all the reply my protein is filgrastim and is biosimilar to
Neupogen. it is stable at acidic pH of 4.0. i want to get rid of dimer
before i formulate it as we will be maintaining it in liquid form. What i
understand TCEP wont work. if i have to use SEC what buffer should i use. My
resin is Superdex 75 prep grade and i am using 10 mM Na Acetate buffer
containing 150 mM NaCl pH 4.0 for SEC.

Once again thanks for all your replies.


On 3/26/10, Ho Leung Ng <[email protected]> wrote:
>
> Does your SDS-PAGE loading buffer contain a reducing agent like beta
> mercaptoethanol? That could be responsible for the difference between
> your SDS-PAGE and HPLC results.
>
>
> ho
>
> On Fri, Mar 26, 2010 at 5:01 PM, CCP4BB automatic digest system
> <[email protected]> wrote:
> > There are 5 messages totaling 490 lines in this issue.
> >
> > Topics of the day:
> >
> >  1. TCEP effect on protein (4)
> >  2. 3 PhD studentships available immediately
> >
> > ----------------------------------------------------------------------
> >
> > Date:    Thu, 25 Mar 2010 22:51:30 -0800
> > From:    megha goyal <[email protected]>
> > Subject: TCEP effect on protein
> >
> > Hi all,
> >
> > My protein is relatively pure except the dimer. i used 10 mM TCEP to
> reduce
> > it (directly added 1 M TCEP to make final volume of 10mM and kept at room
> > temperature for 10 mins] then i dialysed the protein sample to remove
> TCEP
> > [dialysis buffer is Na acetate pH 4.0].
> >
> > On performing SDS PAGE analysis after dialysis of the protein we are
> getting
> > no dimer band, only band of our protein is observed and same is the case
> > with UV reading there is no change in it. But the HPLC analysis of the
> > protein shows two peaks instead of one peak as observed before TCEP
> > treatment. what can be the reason for this. Kindly guide. i need the
> protein
> > to formulate and conduct stability studies on the sample. the protein we
> > obtain after IEX is pure except the dimer and i do not want to go for SEC
> as
> > it greatly reduces protein content and also is quite time consuming. any
> > light on what is happening will bevery useful.
> >
> > thanks and regards
> >
> > ------------------------------
> >
> > Date:    Fri, 26 Mar 2010 08:37:43 +0100
> > From:    Ganesh Natrajan <[email protected]>
> > Subject: Re: TCEP effect on protein
> >
> >
> >
> > Hi Megha,
> >
> > The two peaks on the HPLC indicate that your protein is
> > existing in a monomer-dimer equilibrium in solution. The dimerisation is
> > most probably caused by disulphide bridges. The use of TCEP is breaking
> > those disulphides and that is causing the equilibrium to move towards the
> > monomeric state. However, when the TCEP is dialysed out, the disulphides
> > start forming again and this is causing the equilibrum to move towards
> the
> > dimeric state, a process clearly hastened by the strongly oxidising pH 4
> of
> > the dialysis buffer.
> >
> > Now it all depends on what you want to do. If you
> > want to use the protein in a (largely) monomeric form, I would recommend
> > that you don't dialyse out the TCEP.
> >
> > regards
> >
> > Ganesh
> >
> >
> > **********************************************
> > Blow, blow, thou winter
> > wind
> > Thou art not so unkind
> > As man's ingratitude;
> > Thy tooth is not so
> > keen,
> > Because thou art not seen,
> > Although thy breath be rude.
> >
> > -William
> > Shakespeare
> > **********************************************
> >
> > On Thu, 25 Mar
> > 2010 22:51:30 -0800, megha goyal  wrote:  Hi all,   My protein is
> > relatively pure except the dimer. i used 10 mM TCEP to reduce it
> (directly
> > added 1 M TCEP to make final volume of 10mM and kept at room temperature
> > for 10 mins] then i dialysed the protein sample to remove TCEP [dialysis
> > buffer is Na acetate pH 4.0].   On performing SDS PAGE analysis after
> > dialysis of the protein we are getting no dimer band, only band of our
> > protein is observed and same is the case with UV reading there is no
> change
> > in it. But the HPLC analysis of the protein shows two peaks instead of
> one
> > peak as observed before TCEP treatment. what can be the reason for this.
> > Kindly guide. i need the protein to formulate and conduct stability
> studies
> > on the sample. the protein we obtain after IEX is pure except the dimer
> and
> > i do not want to go for SEC as it greatly reduces protein content and
> also
> > is quite time consuming. any light on what is happening will bevery
> useful.
> >  thanks and regards
> >
> > --
> >
> > ------------------------------
> >
> > Date:    Fri, 26 Mar 2010 08:49:55 +0100
> > From:    Matthias Zebisch <[email protected]>
> > Subject: Re: TCEP effect on protein
> >
> > Hi Ganesh and Mega!
> >
> > I do not agree with Ganesh. I assume, Megha, that truly reversed
> > phaseHPLC was used. This is a denaturing method and the natural
> > disulfide should not form again during the run.
> > Also pH 4 can not be described "oxidizing". Actually, reduced proteins
> > are often dialyzed against acidic buffers to prevent disulfide formation
> > via the thiolate anion.
> > Still, a reducing agent may be used during the run?
> >
> > Sorry that I can not offer a solution to the real problem. More
> > experimental details may be necessary.
> >
> > Bets regards, Matthias
> >
> > Am 3/26/2010 8:37 AM, schrieb Ganesh Natrajan:
> >>
> >> Hi Megha,
> >>
> >> The two peaks on the HPLC indicate that your protein is existing in a
> >> monomer-dimer equilibrium in solution. The dimerisation is most
> >> probably caused by disulphide bridges. The use of TCEP is breaking
> >> those disulphides and that is causing the equilibrium to move towards
> >> the monomeric state. However, when the TCEP is dialysed out, the
> >> disulphides start forming again and this is causing the equilibrum to
> >> move towards the dimeric state, a process clearly hastened by the
> >> strongly oxidising pH 4 of the dialysis buffer.
> >>
> >> Now it all depends on what you want to do. If you want to use the
> >> protein in a (largely) monomeric form, I would recommend that you
> >> don't dialyse out the TCEP.
> >>
> >> regards
> >>
> >> Ganesh
> >>
> >> **********************************************
> >> Blow, blow, thou winter wind
> >> Thou art not so unkind
> >> As man's ingratitude;
> >> Thy tooth is not so keen,
> >> Because thou art not seen,
> >> Although thy breath be rude.
> >>
> >> -William Shakespeare
> >> **********************************************
> >>
> >> On Thu, 25 Mar 2010 22:51:30 -0800, megha goyal <[email protected]>
> >> wrote:
> >>
> >>     Hi all,
> >>     My protein is relatively pure except the dimer. i used 10 mM TCEP
> >>     to reduce it (directly added 1 M TCEP to make final volume of 10mM
> >>     and kept at room temperature for 10 mins] then i dialysed the
> >>     protein sample to remove TCEP [dialysis buffer is Na acetate pH
> 4.0].
> >>     On performing SDS PAGE analysis after dialysis of the protein we
> >>     are getting no dimer band, only band of our protein is observed
> >>     and same is the case with UV reading there is no change in it. But
> >>     the HPLC analysis of the protein shows two peaks instead of one
> >>     peak as observed before TCEP treatment. what can be the reason for
> >>     this. Kindly guide. i need the protein to formulate and conduct
> >>     stability studies on the sample. the protein we obtain after IEX
> >>     is pure except the dimer and i do not want to go for SEC as it
> >>     greatly reduces protein content and also is quite time consuming.
> >>     any light on what is happening will bevery useful.
> >>     thanks and regards
> >>
> >> --
> >>
> >
> >
> > --
> > ****************************************************
> > Dr. Matthias Zebisch
> > Universität Leipzig
> > Biotechnologisch-Biomedizinisches Zentrum
> > Strukturanalytik von Biopolymeren
> > Deutscher Platz 5
> > 04103 Leipzig
> > Germany
> > Phone: 0049-341-97-31323 (lab) -31312 (office)
> > Fax  : 0049-341-97-31319
> > email: [email protected]
> > ****************************************************
> >
> > ------------------------------
> >
> > Date:    Fri, 26 Mar 2010 10:53:07 +0000
> > From:    "Hough, Mike" <[email protected]>
> > Subject: 3 PhD studentships available immediately
> >
> > Dear CCP4bb,
> >
> > The following three studentship positions are available immediately at
> the University of Liverpool. Could you please pass these details on to any
> students in your departments or elsewhere who may be interested? Replies to
> the email addresses listed below, rather than to me please.
> >
> > Thanks,
> >
> > Mike
> >
> >
> > School of Biological Sciences, University of Liverpool
> >
> > 4-year joint BBSRC PhD Studentships – applications invited immediately
> >
> > Three PhD studentships are available in the Molecular Biophysics Group
> for research in the area of x-ray structural biology using the most advanced
> synchrotron radiation sources and the new light sources in the form of x-ray
> free electron lasers (XFELs). The studentships involve collaborations with
> scientists at the DIAMOND Light Source, UK and at the RIKEN Spring-8 Center,
> Japan. The successful candidates will have the exciting opportunity of
> spending up to 2 years at these premier science facilities working at the
> leading edge of structural biology. We are looking for applications now from
> highly committed and motivated graduates from any of the natural sciences
> who are ordinarily resident in the UK. Contact details and links to detailed
> project descriptions are given below:
> >
> > “Long wavelength X-ray diffraction experiments for structural studies
> from biological redox systems”
> > [Strange, UoL & Wagner, DIAMOND]
> > see: http://www.biophysics.liv.ac.uk/PhD_DLS.pdf
> > contact [email protected]
> >
> > “Metalloproteomics: Structure and function studies of metalloproteins of
> biomedical importance”
> > [Hasnain, UoL & Shiro, RIKEN]
> > see: http://www.biophysics.liv.ac.uk/PhD_RIKEN_Metalloprotein.pdf
> > contact: [email protected]
> >
> > “New Science exploration from XFEL: A new paradigm for structural
> visualisation of macromolecules”
> > [Grossmann, UoL & Ishikawa, RIKEN]
> > see: http://www.biophysics.liv.ac.uk/PhD_RIKEN_XFEL.pdf
> > contact: [email protected]
> >
> > ------------------------------
> >
> > Date:    Fri, 26 Mar 2010 09:40:48 -0700
> > From:    James Holton <[email protected]>
> > Subject: Re: TCEP effect on protein
> >
> > Yes, it is possible that the disulfide is just re-forming when the TCEP
> > is gone.  pH 4 is not favorable for the oxidation, but does not prohibit
> > it either.  Especially if there are traces of metal ions around.  I
> > learned this the hard way, as trace metals can catalyze the oxidation of
> > methionine and selenomethionine as well.  In my hands, adding a pinch of
> > EDTA (~1 mM final conc.) to the fraction coming off the HPLC stabilized
> > the reduced species.  Since the HPLC I was using at the time was made of
> > metal (and showed signs of rust around some of the fittings), it is
> > perhaps not surprising that I had a few ppm of Fe++ in the mobile phase.
> >
> > -James Holton
> > MAD Scientist
> >
> > megha goyal wrote:
> >> Hi all,
> >>
> >> My protein is relatively pure except the dimer. i used 10 mM TCEP to
> >> reduce it (directly added 1 M TCEP to make final volume of 10mM and
> >> kept at room temperature for 10 mins] then i dialysed the protein
> >> sample to remove TCEP [dialysis buffer is Na acetate pH 4.0].
> >>
> >> On performing SDS PAGE analysis after dialysis of the protein we are
> >> getting no dimer band, only band of our protein is observed and same
> >> is the case with UV reading there is no change in it. But the HPLC
> >> analysis of the protein shows two peaks instead of one peak as
> >> observed before TCEP treatment. what can be the reason for this.
> >> Kindly guide. i need the protein to formulate and conduct stability
> >> studies on the sample. the protein we obtain after IEX is pure except
> >> the dimer and i do not want to go for SEC as it greatly reduces
> >> protein content and also is quite time consuming. any light on what is
> >> happening will bevery useful.
> >>
> >> thanks and regards
> >
> > ------------------------------
> >
> > End of CCP4BB Digest - 25 Mar 2010 to 26 Mar 2010 (#2010-82)
> > ************************************************************
> >
>

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